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Organized by:
PhysChem Forum Committee and Medicinal Chemistry and Pharmaceutical Technology Subcommittee of the Hungarian Academy of Sciences
The PhysChem Forum Committee are pleased to announce our twelfth Physical Chemistry Forum will be held at the Hungarian Academy of Sciences (HAS), Main building, Budapest, Hungary on Thursday 19th April 2012.
This symposium will have the themes: design of lead molecules with more appropriate physico-chemical properties; models of gastro-intestinal absorption; special issues of solubility and dissolution measurements and new applications of PAMPA method.
The programme will comprise a mixture of presentations and posters with ample opportunity dedicated to questions.
The speakers will be include: Paul Leeson (GSK), keynote; György Keserű (Gedeon Richter); Nathalie Gobeau (Novartis); Andy Davis (AstraZeneca); Edmund Kostewicz (Geothe University); Joerg Berghausen (Novartis); György Balogh (Gedeon Richter); Bálint Sinkó (Semmelweis University)
All posters are welcome but the presentations are reserved for non-commercial work. A prize, kindly sponsored by Sirius Analytical will be awarded to the best poster as dedicated by the committee.
We shall be holding a "Welcome Dinner", including a keynote presentation by Paul Leeson at Hotel President Budapest, on 18th April 2012 (the evening before the symposium).
Fifty rooms have been reserved at the hotel for delegates. If, you would like a room please advise us using the registration form and a booking will be made on your behalf – on a first come first served bases.
Please note the cost of the pre-symposium dinner is € 40 (VAT and drinks included) and this will need to be paid upon arrival along with the delegate room rate of € 99 (single room) or € 109 (double room), which includes buffet-breakfast and all relevant taxes.
If you would like to attend the dinner and the keynote talk without staying at the hotel, payment for dinner would be required at registration at the hotel on 18th April.
There is no registration fee for this meeting, registration is now CLOSED.
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Welcome Dinner, Wednesday 18th April 2012 At the Hotel President, Budapest |
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18.00 – 19.00 |
Registration, Welcome drink |
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19.00 – 19.45 |
Keynote Lecture: Impact of physicochemical properties on drug design Paul Leeson (GSK) |
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20.15 - |
Symposium Dinner |
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Symposium Program, Thursday 19th April 2012 At the building of Hungarian Academy of Sciences, Main Lecture Hall |
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8.30 – 9.00 |
Late Registration |
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Morning session |
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9.00 – 9.20 |
Welcome Krisztina Takács-Novák (chair of local Organising Committee) István Greiner (president of Medicinal Chemistry Subcommittee of HAS) Antonio Llinŕs (member of PhysChem Forum Committee) |
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Chair: Antonio Llinŕs (Astra Zeneca) |
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9.20 – 10.00 |
Medicinal chemistry optimizations – the case for Nature and Nurture György Keserű (Gedeon Richter) |
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10.00 – 10.40 |
Building hypotheses using PBPK modeling Nathalie Gobeau (Novartis) |
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Coffee and Posters |
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Chair: Karl Box (Sirius Analyticals) |
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11.00 – 11.40 |
Impact of gastro-intestinal precipitation on oral drug absorption Edmund Kostewicz (Geothe University, Frankfurt) |
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Lunch and Posters |
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Afternoon session – Chair: Klara Valko (GSK) |
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13.40 – 14.20 |
Physico-chemical properties – the chemist’s contribution to formulation development Joerg Berghausen (Novartis) |
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14.20 - 15.00 |
The key to controlling Compound quality through QSARs Andy Davis (AstraZeneca) |
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15.00 – 15.10 |
Best Poster Prize |
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Coffee and Posters |
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Chair: István Greiner (Gedeon Richter) |
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15.40 – 16.00 |
Skin-PAMPA, a new method for fast prediction of skin permeability Bálint Sinkó (Semmelweis University) |
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16.00 – 16.20 |
Grad-PAMPA based in vitro assay for drug-induced phospholipidosis in early stage of drug discovery György Balogh (Gedeon Richter) |
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16.20 – 16.30 |
Closing the symposium |
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Departure |
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The organizers keep the right to make changes on the preliminary program.
Participants can reach the main building of HAS walking (8-10 min). Organisers will be waiting at the hotel hall and will guide the participants to the Academy. Click here to see a map of the route.
Hotel President, Budapest (H-1054 Budapest, Hold str. 3-5. Tel: +36-1-472-0480)
Directions to the hotel can be found at: http://www.hotelpresident.hu
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A pre-symposium workshop titled: “logP and pKa property prediction and training by ChemAxon technology” organized by ChemAxon Ltd. on 18th April, 16.30-17.30 at Hotel President Budapest. For more information and registration please contact: http://www.chemaxon.com/events/chemaxon-workshop-on-physchem-forum/
For delegates who will stay an extra day in Budapest a one-day post-symposium tour is organized on Friday, 20th April by Yourways Ltd. It will commence at 8.30 am at the Hotel and will end at 18.00 (at the latest) back at the Hotel. Click here to see details.
Chemical Works of Gedeon Richter
EGIS Pharmaceuticals
TEVA
Sirius Analyticals
Heath Scientific
ChemAxon
MestreNova
Paraytec 
